166108-71-0 Fmoc-AEEA-OH shine mai haɗin ADC mai sassauƙa wanda aka yi amfani dashi a cikin haɗin haɗin magungunan antibody-magunguna (ADCs).Fmoc-8-amino-3,6-dioxaoctanoic acid kuma shine mai haɗin PROTAC na tushen PEG wanda za'a iya amfani dashi a cikin haɗin PROTACs.
166108-71-0 Fmoc-AEEA-OH kuma na iya zama ɗaya daga cikin Semaglutide Intermediates.
Babban tasirin semaglutide shine kula da nau'in ciwon sukari na 2 ta hanyar rage matakan glucose na jini.Yana yin kwaikwayon insulin-kamar peptide-1 hormone, wanda ke motsa ƙwayar insulin kuma yana hana sakin glucagon, don haka rage matakan glucose na jini.Semaglutide baya ba da gudummawa ga haɗarin hypoglycemia na faruwa idan aka kwatanta da maganin insulin na al'ada saboda tsarin aikinsa ya fi rikitarwa kuma daidai.Ta hanyar daidaita ma'auni na insulin da glucagon, somalutide zai iya taimaka wa masu fama da ciwon sukari na 2 mafi kyawun sarrafa matakan sukarin jini.
Baya ga rage matakan sukari na jini, semaglutide kuma na iya rage nauyin jiki.Wannan ya faru ne saboda tasirin sa na cin abinci.semaglutide yana motsa ayyukan cibiyar satiety a cikin hypothalamus, wanda ke rage ci.Babban fa'idar semaglutide akan sauran magungunan asarar nauyi shine cewa yana rasa nauyi yayin inganta juriya na insulin da sarrafa sukarin jini.Wannan ya sa ya zama kyakkyawan zaɓi na magani ga marasa lafiya masu ciwon sukari tare da kiba.
Bugu da ƙari, semaglutide yana inganta aikin pancreatic kuma yana rage martanin kumburi a cikin ƙwayoyin islet na pancreatic.Yana kare ƙwayoyin tsibiri daga ƙarin lalacewar da ciwon sukari ke haifarwa kuma yana haɓaka haɓakar ƙwayoyin tsibiri.Wannan yana da mahimmanci musamman ga mutanen da ke da nau'in ciwon sukari na 2, saboda yawan lalacewar ƙwayoyin tsibiri na iya haifar da gazawar tsibiri.
Gabaɗaya, semaglutide magani ne mai inganci kuma mai aminci don maganin nau'in ciwon sukari na 2.Yana taimaka wa marasa lafiya mafi kyawun sarrafa ciwon sukari da rage rikice-rikice ta hanyar rage matakan glucose na jini, rage nauyin jiki, haɓaka aikin tsibiri, da kare ƙwayoyin tsibiri.Nazarin gaba zai kara gano yuwuwar somatostatin a cikin maganin wasu cututtuka, irin su NAFLD da kiba.